Search results for "PEG 400"

showing 5 items of 5 documents

PEG 400/Cerium Ammonium Nitrate Combined with Microwave-Assisted Synthesis for Rapid Access to Beta-Amino Ketones. An Easy-to-Use Protocol for Discov…

2018

Compound libraries are important requirement in target-based drug discovery. In the present work, a small focused compound library based on β-aminoketone scaffold has been prepared combining microwave-assisted organic synthesis (MAOS) with polymer-assisted solution phase synthesis (PASPS) and replacing reaction workup standard purification procedures with solid phase extraction (SPE). Specifically, the effects of solvent, such as dioxane, dimethylformamide (DMF), polyethylene glycol 400 (PEG 400), temperature, irradiation time, stoichiometric ratio of reagents, and catalysts (HCl, acetic acid, cerium ammonium nitrate (CAN)) were investigated to maximize both conversion and yield. The optimi…

3003Transcription FactorPharmaceutical ScienceNitratePolyethylene Glycol01 natural sciencesPolyethylene GlycolsPolymer-assisted solution phase synthesiAnalytical Chemistrychemistry.chemical_compoundDrug DiscoveryMannich reactionSolid phase extractionMicrowavesβ-aminoketonesCeriumKetonesKetoneDNA-Binding ProteinsSolventCeriumChemistry (miscellaneous)Molecular MedicineDimethylformamideMicrowave-assisted organic synthesiMannich reaction; β-aminoketones; microwave-assisted organic synthesis; polymer-assisted solution phase synthesis; solid phase extraction; drug discoveryDNA-Binding ProteinBacterial Proteinchemistry.chemical_elementPolyethylene glycol010402 general chemistryArticlelcsh:QD241-441Bacterial Proteinslcsh:Organic chemistryΒ-aminoketonePhysical and Theoretical ChemistrySolid phase extractionpolymer-assisted solution phase synthesisPEG 400Nitrates010405 organic chemistryDrug Discovery3003 Pharmaceutical ScienceOrganic ChemistrySettore CHIM/08 - Chimica FarmaceuticaCombinatorial chemistry0104 chemical scienceschemistryYield (chemistry)microwave-assisted organic synthesisOrganic synthesisMicrowaveTranscription FactorsMolecules
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Solubilisation of multi walled carbon nanotubes by alpha-pyrene functionalised PMMA and their liquid crystalline self-organisation.

2008

alpha-Pyrene functionalised poly(methyl methacrylate) (PMMA) chains were synthesised by RAFT polymerisation and found to be highly efficient to solubilise and disentangle multi walled carbon nanotubes that can now self-organise as liquid crystalline phases in PMMA and PEG 400 matrices.

PEG 400Materials scienceLiquid crystallineMetals and AlloysGeneral ChemistryRaftCarbon nanotubeCatalysisSurfaces Coatings and FilmsElectronic Optical and Magnetic Materialslaw.inventionchemistry.chemical_compoundSelf organisationchemistryPolymerizationChemical engineeringlawMaterials ChemistryCeramics and CompositesOrganic chemistryPyreneMethyl methacrylateChemical communications (Cambridge, England)
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Rheological characterization of chitosan matrices: Influence of biopolymer concentration

2007

Viscoelastic properties of chitosan (CH), chitosan-poly(ethylene glycol) 400 (CH-PEG), and chitosan-poly(ethylene glycol) 400 with glyoxal as crosslinking agent (CH-PEG-Gly) systems were studied to analyze the effect of chitosan concentration (from 0.83 to 1.67%). Dynamic moduli increase as chitosan concentration increases for all systems. For CH and CH-PEG systems the loss modulus (G″) is greater than the storage modulus (G′) with predominance of the viscous over the elastic behavior. This corresponds to the characteristic behavior of solutions (nonstructured systems). The presence of PEG 400 induces a complementary reinforcement of the mechanical properties of the system. Except for the l…

PEG 400Materials sciencePolymers and PlasticsRheometrytechnology industry and agricultureConcentration effectmacromolecular substancesGeneral ChemistryDynamic mechanical analysisViscoelasticitySurfaces Coatings and Filmschemistry.chemical_compoundChemical engineeringchemistryDynamic modulusMaterials ChemistryGlyoxalComposite materialEthylene glycolJournal of Applied Polymer Science
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Crystallization and preliminary X-ray analysis of native and selenomethionyl vinorine synthase from Rauvolfia serpentina.

2005

Vinorine synthase (VS) is a central enzyme of the biosynthesis of the antiarrhythmic drug ajmaline and is a member of the BAHD superfamily of acyltransferases. So far, no three-dimensional structure with significant sequence homology with VS is known. Crystals of VS and selenomethionyl-labelled VS from the medicinal plant Rauvolfia serpentina have been obtained by the hanging-drop technique at 305 K with ammonium sulfate and PEG 400 as precipitants. VS crystals diffract to 2.8 Å and belong to space group P212121, with unit-cell parameters a = 82.3, b = 89.6, c = 136.2 Å. The selenomethionyl VS crystal was nearly isomorphous with the VS crystal.

StereochemistryCrystallography X-RayRauwolfialaw.inventionIndole AlkaloidsLigaseschemistry.chemical_compoundBiosynthesisStructural BiologylawRauvolfia serpentinamedicineCrystallizationSelenomethioninePlant ProteinsPEG 400chemistry.chemical_classificationATP synthasebiologyGeneral Medicinebiology.organism_classificationAjmalineEnzymechemistryAcyltransferasesbiology.proteinCrystallizationmedicine.drugActa crystallographica. Section D, Biological crystallography
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Determining the selective impregnation of waterlogged archaeological woods with poly(ethylene) glycols mixtures by differential scanning calorimetry

2012

The differential scanning calorimetry (DSC) technique was demonstrated to be a reliable and fast tool for the investigation of the selective impregnation of archaeological woods with poly(ethylene) glycols (PEGs) mixtures. To this aim, waterlogged archaeological woods were impregnated by using aqueous mixtures of PEG 4000 and PEG 400 as well as mixtures of these polymers in the melt state. The efficiency of the treatments was also estimated by determining the total consolidant content entrapped into the cavities of degraded wood by means of DSC and thermogravimetry.

chemistry.chemical_classificationPEG 400EthyleneMaterials scienceAqueous solutiontechnology industry and agriculturemacromolecular substancesPolymerCondensed Matter PhysicsArchaeologyThermogravimetryCultural Heritage Woodchemistry.chemical_compoundDifferential scanning calorimetrychemistryPEG ratioPhysical and Theoretical ChemistryPoly ethyleneSettore CHIM/02 - Chimica Fisica
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